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CAS No.79517-01-4 | Octreotide

Name: Octreotide CAS No.79517-01-4 MF:C51H70N10O12S2 MW:1079.3 Purity:98% Package:1g,25g,50g,100g,250g Worldwide Delivery

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Biochemicals

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Product introduction

Introduction and application of CAS No. 79517-01-4 | Octreotide

Synonyms:SMS-201-995;

OCTREOTIDE(SMS201-995),ACETATE;

cyclic(2-7)-disulfide,(r-l-threonyl-n-(2-hydroxy-1-(hydroxymethyl)propyl);

Octreotide(D-Phe5,Cys6·11,D-Trp8,L-Threoninol12)-SoMatostatin-14(5-12),SMS-201-995;

D-Phenylalanyl-L-cysteinyl-L-phenylalanyl-D-tryptophyl-L-lysyl-L-threonyl-N-[(1R,2R)-2-hydroxy-1-(hydroxyMethyl)propyl]-;

D-Phe-Cys-Phe-D-Trp-Lys-Thr-Cys-Threoninol(DisulfidebridgeCys2-Cys7)

Specification:

ITEMS	SPECIFICATION
CAS	79517-01-4
MF	C51H70N10O12S2
MW	1079.3
Melting point	153-156°C
Color	White to off white
Solubility	soluble in water
Form	Solid
Storage condition	Inert atmosphere,Store in freezer, under -20°C

Digestive system medications:

Octreotide is a digestive system drug. It is a synthetic octapeptide cyclic compound. It is a homolog of natural somatostatin. It has the pharmacological activity of natural somatostatin and has long-acting effects (the half-life of this product is 1.5 hours, compared with 2 to 3 minutes for natural somatostatin). This product has a selective inhibitory effect on the secretion of growth hormone, glucagon and insulin, and is stronger than natural somatostatin. It has been proven by animal experiments: intravenously injecting this product for 15 minutes will inhibit the release of growth hormone as much as natural growth. It is 70 times stronger than statin, and its inhibitory effect on insulin is 3 times stronger than natural somatostatin. It also has inhibitory effects on thyrotropin, adrenocorticotropic hormone, gastrin, cholecystokinin, and intestinal vasoactive polypeptide, and can inhibit the secretion of gastric acid, pancreatic amylase, lipase, and pepsin. It can slow down the transit time of the gastrointestinal tract, promote the absorption of water and electrolytes, have a constrictive effect on splanchnic blood vessels, reduce splanchnic blood flow, reduce liver blood flow, reduce portal pressure and portal blood flow, and reduce intestinal hyperplasia Secretion, and can enhance intestinal absorption of water and Na+.

Biological activity:

Octreotide acetate is a long-acting synthetic analog of natural somatostatin and a more potent inhibitor of growth hormone, glucagon and insulin than somatostatin.

Package and transportation :

Package: 10g,25g,50g,100g,250g